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Imidazole[5,1-f][1,2,4]triazin-4(3H)-one

  Vardenafil core synthesis.

Pyrazolo[4,3-d]pyrimidin-7-one

  Sildenafil core structure, the cycylization need to use H2O2 in EtOH

From aminopyridine:

   
   
   

 

   

 


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